5-Membered Heterocycle Synthesis Using Iodine
- 1st Edition - January 24, 2023
- Imprint: Elsevier
- Author: Navjeet Kaur
- Language: English
- Paperback ISBN:9 7 8 - 0 - 4 4 3 - 1 8 9 4 1 - 8
- eBook ISBN:9 7 8 - 0 - 4 4 3 - 1 8 9 4 2 - 5
5-Membered Heterocycle Synthesis Using Iodine presents both old and new methods for the synthesis of various five-membered heterocycles using iodine, providing information for ma… Read more
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Request a sales quote5-Membered Heterocycle Synthesis Using Iodine presents both old and new methods for the synthesis of various five-membered heterocycles using iodine, providing information for making specific compounds using particular reagents. Heterocyclic frameworks represent the main structural subunits of many biologically active compounds and natural products, and the ability of heterocycles to act both as reactive pharmacophores and biomimetics has greatly contributed to their unique value as traditional key elements of various drugs. Contemporary developments in process chemistry and discovery emphasize novel sustainable synthetic pathways as fast and ecologically acceptable alternatives to the traditional protocols.
This book serves as a guide for students, pharmacologists, biochemists, organic and medicinal chemists, researchers, and academic professionals to obtain easy access to synthetic protocols for different five-membered heterocycles using iodine.
- Covers the applications of five-membered heterocycles
- Highlights methodologies for the synthesis of five-membered heterocycles using iodine
- Contains the most up-to-date information in this fast-moving field
Students and Researchers in Chemistry, Synthetic Chemists, Organic Chemists
- Cover image
- Title page
- Table of Contents
- Copyright
- Biography
- Preface
- List of abbreviations
- 1. Five-membered N-heterocycles–Part I
- 1.1. Introduction
- 1.2. Synthesis of pyrroles
- 1.3. Synthesis of indoles
- 1.4. Synthesis of fused five-membered N-heterocycles
- 2. Five-membered N-heterocycles—Part II
- 2.1. Introduction
- 2.2. Synthesis of five-membered N-heterocycles from haloamines
- 2.3. Synthesis of five-membered N-heterocycles from furans
- 3. Five-membered N-heterocycles: cyclization of alkenyl systems
- 3.1. Introduction
- 3.2. Synthesis of five-membered N-heterocycles from alkenes
- 4. Five-membered N-heterocycles: cyclization of alkynyl systems
- 4.1. Introduction
- 4.2. Synthesis of five-membered N-heterocycles from alkynes
- 5. Five-membered N,N-heterocycles
- 5.1. Introduction
- 5.2. Synthesis of pyrazoles
- 5.3. Synthesis of indazoles and fused pyrazoles
- 5.4. Synthesis of imidazoles
- 5.5. Synthesis of benzimidazoles
- 5.6. Synthesis of fused imidazoles
- 6. Five-membered N,N,N- and N,N,N,N-heterocycles
- 6.1. Introduction
- 6.2. Synthesis of triazoles
- 6.3. Synthesis of tetrazoles
- 7. Five-membered O-heterocycles: cyclization of C=C with OH—Part I
- 7.1. Introduction
- 7.2. Synthesis of furans
- 8. Five-membered O-heterocycles: cyclization of CC with OH—Part II
- 8.1. Introduction
- 8.2. Synthesis of benzofurans
- 8.3. Synthesis of fused furans
- 9. Five-membered O-heterocycles: cyclization of alkenyl or alkynyl compounds
- 9.1. Introduction
- 9.2. Synthesis of five-membered O-heterocycles from alkenes
- 9.3. Synthesis of five-membered O-heterocycles from alkynes
- 10. Five-membered O- and O,O-heterocycles
- 10.1. Introduction
- 10.2. Synthesis of furans
- 10.3. Synthesis of benzofurans
- 10.4. Synthesis of fused furans
- 10.5. Synthesis of dioxolanes
- 11. Five-membered O,N-heterocycles
- 11.1. Introduction
- 11.2. Synthesis of isoxazoles
- 11.3. Synthesis of oxazoles
- 11.4. Synthesis of benzoxazoles
- 11.5. Synthesis of fused oxazoles
- 12. Five-membered O,N,N-heterocycles: hydrazine derivatives
- 12.1. Introduction
- 12.2. Synthesis of oxadiazoles from thiosemicarbazides
- 12.3. Synthesis of oxadiazoles from semicarbazones
- 12.4. Synthesis of oxadiazoles from hydrazine derivatives
- 13. Five-membered S-heterocycles
- 13.1. Introduction
- 13.2. Synthesis of thiophenes
- 13.3. Synthesis of benzothiophenes
- 13.4. Synthesis of fused thiophenes
- 13.5. Synthesis of dithiolanes
- 13.6. Synthesis of thiadiazoles
- 14. Five-membered S,N-heterocycles
- 14.1. Introduction
- 14.2. Synthesis of 1,2-thiazoles
- 14.3. Synthesis of 1,3-thiazoles
- 14.4. Synthesis of benzothiazoles
- 14.5. Synthesis of fused thiazoles
- Index
- Edition: 1
- Published: January 24, 2023
- Imprint: Elsevier
- No. of pages: 500
- Language: English
- Paperback ISBN: 9780443189418
- eBook ISBN: 9780443189425
NK
Navjeet Kaur
Dr. Navjeet Kaur received her BSc from Panjab University Chandigarh (Panjab, India) in 2008. In 2010, she completed her MSc in Chemistry from Banasthali Vidyapith. She was awarded with PhD in 2014 by the same university. With 11 years of teaching experience, she has published over 160 scientific research papers, review articles, book chapters, and monographs in the field of organic synthesis in national and international reputed journals. She has published five authored books: with Elsevier. She secured her place amongst top 2% scientists of the world in 2017 (single year ranking), 2018 (full career wise ranking), 2019 [full career wise ranking with 424 world rank (04 in India) and single year ranking with 03 world rank (01 in India)] and 2020 (full career wise ranking with 372 world rank and single year ranking with 126 world rank). In 2021, Dr. Kaur was chosen as a candidate for membership by Royal Society of Research, London, England, UK with full waiver of application fees. She is serving as an Editor-in-Chief of the “Advanced Chemicobiology Research” journal.
Affiliations and expertise
Lovely Professional University, IndiaRead 5-Membered Heterocycle Synthesis Using Iodine on ScienceDirect